Dirk Tourwé

Overview

Best Publications

• "Click to chelate": synthesis and installation of metal chelates into biomolecules in a single step.

  Thomas L. Mindt;Harriet Struthers;Luc Brans;Todor Anguelov

  444
  Citations

• Structural basis for bifunctional peptide recognition at human δ-opioid receptor

  Gustavo Fenalti;Gustavo Fenalti;Nadia A. Zatsepin;Cecilia Betti;Patrick T. Giguere

  204
  Citations

• Effect of temperature on retention of enantiomers of β-methyl amino acids on a teicoplanin chiral stationary phase

  Antal Péter;Gabriella Török;Daniel W Armstrong;Géza Tóth

  191
  Citations

• In vitro and in vivo evaluation of new radiolabeled neurotensin(8–13) analogues with high affinity for NT1 receptors

  Elisa Garcı́a Garayoa;Lesley Allemann-Tannahill;Peter Bläuenstein;Martine Willmann

  134
  Citations

• A 99mTc(I)-postlabeled high affinity bombesin analogue as a potential tumor imaging agent.

  La Bella R;Garcia-Garayoa E;Bahler M;Bläuenstein P

  127
  Citations

• Influence of the molecular charge on the biodistribution of bombesin analogues labeled with the [99mTc(CO)3]-core.

  Elisa García Garayoa;Christian Schweinsberg;Veronique Maes;Luc Brans

  121
  Citations

• Chemical and biological characterization of new Re(CO)3/[99mTc](CO)3 bombesin analogues ☆

  Elisa García Garayoa;Dominique Rüegg;Peter Bläuenstein;Martin Zwimpfer

  112
  Citations

• Biodistribution and catabolism of 18F-labeled neurotensin(8-13) analogs

  Ralf Bergmann;Matthias Scheunemann;Christoph Heichert;Peter Mäding

  112
  Citations

• Conformational restriction of Tyr and Phe side chains in opioid peptides: information about preferred and bioactive side-chain topology.

  Dirk Tourwé;Kris Verschueren;Anne Frycia;Peg Davis

  106
  Citations

• Novel Glycated [99mTc(CO)3]-Labeled Bombesin Analogues for Improved Targeting of Gastrin-Releasing Peptide Receptor-Positive Tumors

  Christian Schweinsberg;Veronique Maes;Luc Brans;Peter Bläuenstein

  98
  Citations

• Preclinical Evaluation of a New, Stabilized Neurotensin(8–13) Pseudopeptide Radiolabeled with 99mTc

  Elisa García-Garayoa;Peter Bläuenstein;Matthias Bruehlmeier;Alain Blanc

  96
  Citations

• Stabilization of neurotensin analogues: effect on peptide catabolism, biodistribution and tumor binding

  Matthias Bruehlmeier;Elisa Garcı́a Garayoa;Alain Blanc;Barbara Holzer

  92
  Citations

• A click approach to structurally diverse conjugates containing a central di-1,2,3-triazole metal chelate.

  Thomas L. Mindt;Christian Schweinsberg;Luc Brans;Adelheid Hagenbach

  83
  Citations

• Beta-homo-amino acid scan of angiotensin IV.

  Aneta Lukaszuk;Heidi Demaegdt;Erzsebet Szemenyei;Géza Tóth

  82
  Citations

• Theoretical study revealing the functioning of a novel combination of catalytic motifs in histone deacetylase.

  K. Vanommeslaeghe;F. De Proft;S. Loverix;D. Tourwé

  80
  Citations

• DFT-based ranking of zinc-binding groups in histone deacetylase inhibitors.

  Kenno Vanommeslaeghe;Stefan Loverix;Paul Geerlings;Dirk Tourwe

  79
  Citations

• Liquid chromatographic study of the enzymatic degradation of endomorphins, with identification by electrospray ionization mass spectrometry.

  Antal Péter;Géza Tóth;Csaba Tömböly;Georges Laus

  77
  Citations

• Novel 99mTc-labeled neurotensin analogues with optimized biodistribution properties.

  Veronique Maes;Elisa Garcia-Garayoa;Peter Bläuenstein;Dirk Tourwé

  75
  Citations

• Comparison of the separation efficiencies of chirobiotic T and TAG columns in the separation of unusual amino acids.

  Antal Péter;Anita Árki;Dirk Tourwé;Enikő Forró

  73
  Citations

• Novel DOTA-neurotensin analogues for 111In scintigraphy and 68Ga PET imaging of neurotensin receptor-positive tumors.

  Faisal Alshoukr;Aurélie Prignon;Luc Brans;Abdelhak Jallane;Abdelhak Jallane;Abdelhak Jallane

  72
  Citations

• High-performance liquid chromatographic separation of the enantiomers of unusual α-amino acid analogues

  Antal Péter;Edit Olajos;Richard Casimir;Dirk Tourwé

  71
  Citations