Marino Artico

Overview

Best Publications

• New Arylthioindoles: Potent Inhibitors of Tubulin Polymerization. 2. Structure−Activity Relationships and Molecular Modeling Studies

  Gabriella De Martino;Michael C. Edler;Giuseppe La Regina;Antonio Coluccia

  445
  Citations

• Arylthioindoles, Potent Inhibitors of Tubulin Polymerization

  Gabriella De Martino;Giuseppe La Regina;Antonio Coluccia;Michael C. Edler

  336
  Citations

• Geometrically and Conformationally Restrained Cinnamoyl Compounds as Inhibitors of HIV-1 Integrase: Synthesis, Biological Evaluation, and Molecular Modeling

  M Artico;R Di Santo;R Costi;E Novellino

  239
  Citations

• Arylthioindole inhibitors of tubulin polymerization. 3. Biological evaluation, structure-activity relationships and molecular modeling studies

  Giuseppe La Regina;Michael C. Edler;Andrea Brancale;Sahar Kandil

  229
  Citations

• Novel Indolyl Aryl Sulfones Active against HIV-1 Carrying NNRTI Resistance Mutations: Synthesis and SAR Studies

  Romano Silvestri;Gabriella De Martino;Giuseppe La Regina;Marino Artico

  220
  Citations

• Design, molecular modeling, synthesis, and anti-HIV-1 activity of new indolyl aryl sulfones. Novel derivatives of the indole-2-carboxamide.

  Rino Ragno;Antonio Coluccia;Giuseppe La Regina;Gabriella De Martino

  210
  Citations

• Antimycobacterial pyrroles: synthesis, anti-Mycobacterium tuberculosis activity and QSAR studies

  Rino Ragno;Garland R Marshall;Roberto Di Santo;Roberta Costi

  190
  Citations

• 2-Sulfonyl-4-chloroanilino Moiety: A Potent Pharmacophore for the Anti-Human Immunodeficiency Virus Type 1 Activity of Pyrrolyl Aryl Sulfones

  Artico M;Silvestri R;Massa S;Loi Ag

  185
  Citations

• Structure-based design, synthesis, and biological evaluation of novel pyrrolyl aryl sulfones: HIV-1 non-nucleoside reverse transcriptase inhibitors active at nanomolar concentrations.

  Marino Artico;Romano Silvestri;Eugenia Pagnozzi;Biancamaria Bruno

  183
  Citations

• 5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3, 4-dihydropyrimidin-4(3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives.

  A. Mai;M. Artico;G. Sbardella;S. Massa

  160
  Citations

• New Pyrrole Inhibitors of Monoamine Oxidase: Synthesis, Biological Evaluation, and Structural Determinants of MAO-A and MAO-B Selectivity

  Giuseppe La Regina;Romano Silvestri;Marino Artico;Antonio Lavecchia

  143
  Citations

• Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, biological activities, and mechanism of action.

  Roberto Di Santo;Roberta Costi;Alessandra Roux;Marino Artico

  126
  Citations

• Antifungal Agents. 11. N-Substituted Derivatives of 1-[(Aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazole: Synthesis, Anti-Candida Activity, and QSAR Studies

  Roberto Di Santo;Andrea Tafi;Roberta Costi;Maurizio Botta

  125
  Citations

• Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase.

  A Mai;G Sbardella;M Artico;R Ragno

  118
  Citations

• 2,6-Bis(3,4,5-trihydroxybenzylydene) derivatives of cyclohexanone: novel potent HIV-1 integrase inhibitors that prevent HIV-1 multiplication in cell-based assays

  Roberta Costi;Roberto Di Santo;Marino Artico;Silvio Massa

  114
  Citations

• Computer-aided design, synthesis, and anti-HIV-1 activity in vitro of 2-alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as novel potent non-nucleoside reverse transcriptase inhibitors, also active against the Y181C variant.

  Rino Ragno;Antonello Mai;Gianluca Sbardella;Marino Artico

  111
  Citations

• Docking and 3-D QSAR studies on indolyl aryl sulfones. Binding mode exploration at the HIV-1 reverse transcriptase non-nucleoside binding site and design of highly active N-(2-hydroxyethyl)carboxamide and N-(2-hydroxyethyl)carbohydrazide derivatives.

  Rino Ragno;Marino Artico;Gabriella De Martino;Giuseppe La Regina

  109
  Citations

• Antifungal agents. 10. New derivatives of 1-[(aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-candida activity, and quantitative structure-analysis relationship studies.

  Andrea Tafi;Roberta Costi;Maurizio Botta;Roberto Di Santo

  101
  Citations

• Synthesis, biological evaluation, and binding mode of novel 1-[2-(diarylmethoxy)ethyl]-2-methyl-5-nitroimidazoles targeted at the HIV-1 reverse transcriptase.

  Romano Silvestri;Marino Artico;Gabriella De Martino;Rino Ragno

  99
  Citations

• Pyrrolnitrin and related pyrroles endowed with antibacterial activities against Mycobacterium tuberculosis

  Roberto Di Santo;Roberta Costi;Marino Artico;Silvio Massa

  92
  Citations