Tiziano Tuccinardi

Best Publications

• The History of Nanoscience and Nanotechnology: From Chemical–Physical Applications to Nanomedicine

  Samer Bayda;Muhammad Adeel;Tiziano Tuccinardi;Marco Cordani

  1834
  Citations

• Discovery of N-hydroxyindole-based inhibitors of human lactate dehydrogenase isoform A (LDH-A) as starvation agents against cancer cells.

  Carlotta Granchi;Sarabindu Roy;Chiara Giacomelli;Marco Macchia

  270
  Citations

• What is the current value of MM/PBSA and MM/GBSA methods in drug discovery?

  Tiziano Tuccinardi

  252
  Citations

• Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6.

  Arduino A. Mangoni;Catherine Guillou;Jean Jacques Vanden Eynde;Christopher Hulme

  230
  Citations

• Application of MM-PBSA Methods in Virtual Screening

  Giulio Poli;Carlotta Granchi;Flavio Rizzolio;Tiziano Tuccinardi

  172
  Citations

• Cannabinoid CB2/CB1 selectivity. Receptor modeling and automated docking analysis.

  Tiziano Tuccinardi;Pier Luigi Ferrarini;Clementina Manera;Gabriella Maria Pia Ortore

  138
  Citations

• Matrix Metalloproteinase Inhibitors: New Challenges in the Era of Post Broad-Spectrum Inhibitors

  Elisa Nuti;Tiziano Tuccinardi;Armando Rossello

  137
  Citations

• Targeting Toxic RNAs that Cause Myotonic Dystrophy Type 1 (DM1) with a Bisamidinium Inhibitor.

  Chun Ho Wong;Lien Nguyen;Jessie Peh;Long M. Luu

  121
  Citations

• CDK inhibitors: from the bench to clinical trials.

  Flavio Rizzolio;Tiziano Tuccinardi;Isabella Caligiuri;Chiara Lucchetti

  116
  Citations

• Former foodstuff products in Tenebrio molitor rearing: effects on growth, chemical composition, microbiological load, and antioxidant status.

  Simone Mancini;Filippo Fratini;Barbara Turchi;Simona Mattioli

  114
  Citations

• Docking-based virtual screening: recent developments.

  Tiziano Tuccinardi

  110
  Citations

• Extensive consensus docking evaluation for ligand pose prediction and virtual screening studies.

  Tiziano Tuccinardi;Giulio Poli;Veronica Romboli;Antonio Giordano

  108
  Citations

• Amber force field implementation, molecular modelling study, synthesis and MMP-1/MMP-2 inhibition profile of (R)- and (S)-N-hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)-3-methylbutanamides.

  Tiziano Tuccinardi;Adriano Martinelli;Elisa Nuti;Paolo Carelli

  106
  Citations

• New 1,8-naphthyridine and quinoline derivatives as CB2 selective agonists

  Clementina Manera;Maria Grazia Cascio;Veronica Benetti;Marco Allarà

  101
  Citations

• Design, synthesis, and biological evaluation of new 1,8-naphthyridin-4(1H)-on-3-carboxamide and quinolin-4(1H)-on-3-carboxamide derivatives as CB2 selective agonists.

  Clementina Manera;Veronica Benetti;M. Paola Castelli;Tiziana Cavallini

  100
  Citations

• The dichotomous role of the glycolytic metabolism pathway in cancer metastasis: Interplay with the complex tumor microenvironment and novel therapeutic strategies.

  Btissame El Hassouni;Carlotta Granchi;Andrea Vallés-Martí;I Gede Putu Supadmanaba

  99
  Citations

• α-Glucosidase and α-Amylase Inhibitors from Arcytophyllum thymifolium

  Luigi Milella;Stella Milazzo;Marinella De Leo;Mariela Beatriz Vera Saltos

  95
  Citations

• The TRPA1 channel mediates the analgesic action of dipyrone and pyrazolone derivatives.

  Romina Nassini;Camilla Fusi;Serena Materazzi;Elisabetta Coppi

  95
  Citations

• The Extra-Virgin Olive Oil Polyphenols Oleocanthal and Oleacein Counteract Inflammation-Related Gene and miRNA Expression in Adipocytes by Attenuating NF-κB Activation.

  Sara Carpi;Egeria Scoditti;Marika Massaro;Beatrice Polini

  92
  Citations

• Proposal of a new binding orientation for non-peptide AT1 antagonists: homology modeling, docking and three-dimensional quantitative structure-activity relationship analysis.

  Tiziano Tuccinardi;Vincenzo Calderone;Simona Rapposelli;Adriano Martinelli

  89
  Citations

• N-Hydroxyindole-based inhibitors of lactate dehydrogenase against cancer cell proliferation

  Carlotta Granchi;Sarabindu Roy;Alessio De Simone;Irene Salvetti

  81
  Citations