Paul J. Reider

Research.com Recognitions

• 2011 - NAS Award for Chemistry in Service to Society, U.S. National Academy of Sciences For his contributions to the discovery and development of numerous approved drugs, including those for treating asthma and for treating AIDS.

Overview

Best Publications

• Oxidation of Primary Alcohols to Carboxylic Acids with Sodium Chlorite Catalyzed by TEMPO and Bleach

  Mangzhu Zhao;Jing Li;Eiichi Mano;Zhiguo Song

  590
  Citations

• A New Planar Chiral Bisphosphine Ligand for Asymmetric Catalysis: Highly Enantioselective Hydrogenations under Mild Conditions

  Philip J. Pye;Kai Rossen;Robert A. Reamer;Nancy N. Tsou

  471
  Citations

• Are heterogeneous catalysts precursors to homogeneous catalysts

  Ian W. Davies;Louis Matty;David L. Hughes;Paul J. Reider

  446
  Citations

• Ullmann diaryl ether synthesis: rate acceleration by 2,2,6,6-tetramethylheptane-3,5-dione.

  Elizabeth Buck;Zhiguo Jake Song;David Tschaen;Peter G Dormer

  394
  Citations

• An improved protocol for the preparation of 3-pyridyl- and some arylboronic acids.

  Wenjie Li;Dorian P. Nelson;Mark S. Jensen;R. Scott Hoerrner

  341
  Citations

• Practical Route to a New Class of LTD4 Receptor Antagonists

  Robert D. Larsen;Edward G. Corley;Anthony O. King;James D. Carroll

  313
  Citations

• Efficient Synthesis of Losartan, A Nonpeptide Angiotensin II Receptor Antagonist

  Robert D. Larsen;Anthony O. King;Cheng Y. Chen;Edward G. Corley

  295
  Citations

• Synthesis of Chiral 2,2'-Bis(diphenylphosphino)-1,1'-binaphthyl (BINAP) via a Novel Nickel-Catalyzed Phosphine Insertion

  Dongwei Cai;Joseph F. Payack;Dean R. Bender;David L. Hughes

  289
  Citations

• A novel chromium trioxide catalyzed oxidation of primary alcohols to the carboxylic acids

  Mangzhu Zhao;Jing Li;Zhiguo Song;Richard Desmond

  265
  Citations

• Practical asymmetric synthesis of Efavirenz (DMP 266), an HIV-1 reverse transcriptase inhibitor

  Michael E. Pierce;Rodney L. Parsons;Lilian A. Radesca;Young S. Lo

  263
  Citations

• Synthesis of alpha-amido ketones via organic catalysis: thiazolium-catalyzed cross-coupling of aldehydes with acylimines.

  Jerry A. Murry;Doug E. Frantz;Arash Soheili;Richard Tillyer

  242
  Citations

• A Novel, Highly Enantioselective Ketone Alkynylation Reaction Mediated by Chiral Zinc Aminoalkoxides

  Lushi Tan;Cheng Yi Chen;Richard D. Tillyer;Edward J.J. Grabowski

  229
  Citations

• Highly diastereoselective reaction of a chiral, non-racemic amide enolate with (S)-glycidyl tosylate. Synthesis of the orally active HIV-1 protease inhibitor L-735,524

  David Askin;Kan K Eng;Kai Rossen;Robert M Purick

  214
  Citations

• Syntheses of Indoles via a Palladium-Catalyzed Annulation between Iodoanilines and Ketones.

  Cheng-yi Chen;David R. Lieberman;Robert D. Larsen;Thomas R. Verhoeven

  207
  Citations

• Efficient Synthesis of NK1 Receptor Antagonist Aprepitant Using a Crystallization-Induced Diastereoselective Transformation†

  Karel M. J. Brands;Joseph F. Payack;Jonathan D. Rosen;Todd D. Nelson

  205
  Citations

• Simple and efficient resolution of l,1′-bi-2-naphthol

  Dongwei Cai;David L. Hughes;Thomas R. Verhoeven;Paul J. Reider

  199
  Citations

• Improved Fischer Indole Reaction for the Preparation of N,N-Dimethyltryptamines: Synthesis of L-695,894, a Potent 5-HT1D Receptor Agonist

  Cheng yi Chen;Chris H. Senanayake;Timothy J. Bill;Robert D. Larsen

  182
  Citations

• Total synthesis of thienamycin: a new approach from aspartic acid

  Paul J. Reider;Edward J.J. Grabowski

  180
  Citations

• Highly regioselective Friedländer annulations with unmodified ketones employing novel amine catalysts: syntheses of 2-substituted quinolines, 1,8-naphthyridines, and related heterocycles.

  Peter G. Dormer;Kan K. Eng;Roger N. Farr;Guy R. Humphrey

  176
  Citations

• An efficient synthesis of LTD4 antagonist L-699,392

  A. O. King;E. G. Corley;R. K. Anderson;R. D. Larsen

  170
  Citations

• New air-stable catalysts for general and efficient suzuki-miyaura cross-coupling reactions of heteroaryl chlorides.

  Unknown

  163
  Citations