Joan Bosch

Overview

Best Publications

• Chiral oxazolopiperidone lactams: versatile intermediates for the enantioselective synthesis of piperidine-containing natural products.

  Carmen Escolano;Mercedes Amat;Joan Bosch

  240
  Citations

• Enantioselective synthesis of piperidine, indolizidine, and quinolizidine alkaloids from a phenylglycinol-derived delta-lactam.

  Mercedes Amat;Núria Llor;José Hidalgo;Carmen Escolano

  195
  Citations

• Synthesis of Enantiopure trans-3,4-Disubstituted Piperidines. An Enantiodivergent Synthesis of (+)- and (−)-Paroxetine

  Mercedes Amat;Joan Bosch;José Hidalgo;Margalida Cantó

  173
  Citations

• A General Synthetic Entry to Strychnos Alkaloids of the Curan Type via a Common 3a-(2-Nitrophenyl)hexahydroindol-4-one Intermediate. Total Syntheses of (±)- and (−)-Tubifolidine, (±)-Akuammicine, (±)-19,20-Dihydroakuammicine, (±)-Norfluorocurarine, (±)-Echitamidine, and (±)-20-Epilochneridine1

  Josep Bonjoch;Daniel Solé;Silvina García-Rubio;Joan Bosch

  154
  Citations

• Palladium(0)-Catalyzed Heteroarylation of 2- and 3-Indolylzinc Derivatives. An Efficient General Method for the Preparation of (2-Pyridyl)indoles and Their Application to Indole Alkaloid Synthesis.

  Mercedes Amat;Sabine Hadida;Grigorii Pshenichnyi;Joan Bosch

  139
  Citations

• Elucidation of the structure of methanopterin, a coenzyme from Methanobacterium thermoautotrophicum, using two-dimensional nuclear-magnetic-resonance techniques.

  Patrick Van Beelen;Alphons P. M. Stassen;Johannes W. G. Bosch;Godfried D. Vogels

  133
  Citations

• Biomimetic Total Synthesis of Ervitsine and Indole Alkaloids of the Ervatamine Group via 1,4-Dihydropyridines

  M.-Lluïsa Bennasar;and Bernat Vidal;Joan Bosch

  127
  Citations

• A new synthetic entry to pentacyclic Strychnos alkaloids. Total synthesis of (.+-.)-tubifolidine, (.+-.)-tubifoline, and (.+-.)-19,20-dihydroakuammicine

  Mercedes Amat;Ana Linares;Joan Bosch

  123
  Citations

• A General Method for the Synthesis of Bridged Indole Alkaloids. Addition of Carbon Nucleophiles to N-Alkylpyridinium Salts

  Joan Bosch;M.-Lluïsa Bennasar

  116
  Citations

• Total Synthesis of Uleine-Type and Strychnos Alkaloids through a Common Intermediate

  Jordi Gracia;Nuria Casamitjana;Josep Bonjoch;Joan Bosch

  106
  Citations

• Enantioselective synthesis of 3,3-disubstituted piperidine derivatives by enolate dialkylation of phenylglycinol-derived oxazolopiperidone lactams.

  Mercedes Amat;Oscar Lozano;Carmen Escolano;Elies Molins

  98
  Citations

• Dynamic kinetic resolution of racemic gamma-aryl-delta-oxoesters. Enantioselective synthesis of 3-arylpiperidines.

  Mercedes Amat;Margalida Cantó;Núria Llor;Carmen Escolano

  97
  Citations

• Identification of new aminoacid amides containing the imidazo[2,1-b]benzothiazol-2-ylphenyl moiety as inhibitors of tumorigenesis by oncogenic Met signaling.

  Alessandro Furlan;Francesco Colombo;Andrea Kover;Nathalie Issaly

  97
  Citations

• Conjugate addition of organocuprates to chiral bicyclic delta-lactams. Enantioselective synthesis of cis-3,4-disubstituted and 3,4,5-trisubstituted piperidines.

  Mercedes Amat;Maria Pérez;Núria Llor;Joan Bosch

  92
  Citations

• Total Synthesis of (-)-Strychnine via the Wieland-Gumlich Aldehyde

  Daniel Solé;Josep Bonjoch;Silvina García-Rubio;Emma Peidró

  90
  Citations

• Enantioselective total synthesis of Wieland-Gumlich aldehyde and (-)-strychnine

  Daniel Solé;Josep Bonjoch;Silvina García-Rubio;Emma Peidró

  90
  Citations

• Chiral precursors for the synthesis of enantiomerically pure piperidines. Total synthesis of (R)-(-)-coniine

  Mercedes Amat;Núria Llor;Joan Bosch

  89
  Citations

• Studies on the Synthesis of Strychnos Indole Alkaloids. Synthesis of (.+-.)-Dehydrotubifoline

  Josep Bonjoch;Daniel Sole;Joan Bosch

  88
  Citations

• Preparation and reactions of 1-(tert-butyldimethylsilyl)-3-lithioindole. Regioselective synthesis of 3-substituted indoles

  Mercedes Amat;Sabine Hadida;Swargam Sathyanarayana;Joan Bosch

  85
  Citations

• Conjugate additions to phenylglycinol-derived unsaturated δ-lactams. Enantioselective synthesis of uleine alkaloids

  Mercedes Amat;Maria Perez;Nuria Llor;Carmen Escolano

  82
  Citations

• Enantioselective Synthesis of Indole Alkaloids from Chiral Lactams

  Mercedes Amat;Maria Pérez;Joan Bosch

  80
  Citations

• Cooperative Catalysis for the First Asymmetric Formal [3+2] Cycloaddition Reaction of Isocyanoacetates to α,β‐Unsaturated Ketones

  Carlos Arróniz;Alberto Gil‐González;Vladislav Semak;Carmen Escolano

  75
  Citations